Publications
37. C. Stathakis, P. L. Gkizis, A. L. Zografos, "Metal-catalyzed cycloisomerization as a powerful tool in the synthesis of complex sesquiterpenoids" Nat. Prod. Rep. 2016, 33, 1093.
36. V. P. Demertzidou, A. L. Zografos, "Platinum-catalyzed cycloisomerizations of a common enyne: a divergent entry to cyclopropane sesquiterpenoids" Org. Biomol. Chem. 2016, 14, 6942.
35. S Katsamakas, A. L. Zografos, V. Sarli "Advances of Phenoxazines: Synthesis, Reactivity and Their Medicinal Applications" Curr. Med. Chem. 2016, 23, 2972.
34. "From Biosynthesis to Total Synthesis" Editor: Alexandros Zografos, May 2016, Wiley Hoboken, ISBN: 978-1-118-75173-2
33. T. Katsina, E. E. Anagnostaki, F. Mitsa, V. Sarli, A. L. Zografos " Palladium-Catalyzed Direct Alkenylation of 4-Hydroxy-2-pyridones" RSC Advances, 2016, 6, 6978.
32. E. Kontogiannidou, D. A. Andreadis, A. L. Zografos, H. Nazar, P. Klepetsanis, S. M. van der Merwe, D. G. Fatouros "Ex vivo buccal drug delivery of ropinirole hydrochloride in the precence of permeation enhancers: the effect of charge" Pharm. Develop. Technol. 2016, accepted.
31. E. E. Anagnostaki, V. Demertzidou, A. L. Zografos "Divergent Pathways to Furosesquiterpenes. First Total Syntheses of (+)-Zedoarol and (Rac)-Gweicurculactone" Chem. Comm. 2015, 51, 2364.
30. M. Kalyva, A. L. Zografos, E. Kapourani, E. Giombazolias, L. Devel, A. Papakyriakou, V. Dive, Y. G. Lazarou, D. Georgiadis "Probing the Mechanism of Morita Baylis Hillman Acetates' (MBHAs) Allylic Substitution by Using the Silyl Phosphonite Paradigm: Scope and Applications of a Versatile transformation" Chem.-Eur. J. 2015, 21, 3278.
29. E. E. Anagnostaki, A. D. Fotiadou, V. Demertzidou, A. L. Zografos " Palladium Catalyzed C-3 Arylation of 4-hydroxy-2-Pyridones" Chem. Commun. 2014, 50, 6879.
28. E. Anagnostaki, A. L. Zografos " Furanogermenone as a Stepping Stone for the Synthesis of Various Sesquiterpenoids" Org. Lett. 2013, 15, 152
27. A. Fotiadou, A. L. Zografos "Evidencing Reversibility in 6π-Electrocyclization Reaction. Synthesis of Pyranopyridones" Org. Lett. 2012, 14, 5664
26. A. L. Zografos "Quinolines and Isoquinolines" Heterocyclic Chemistry in Drug Discovery; Chapter 11; Editor: J. J. Li; Wiley & Sons 2012
25. E. Anagnostaki, A. L. Zografos "Common Synthetic Scaffold in the Total Synthesis of Diverse Natural Products" Chem. Soc. Rev. 2012, 41, 5613
24. A. D. Fotiadou, A. L. Zografos "Accesing the structural diversity of pyridone alkaloids: Concise Total Synthesis of Rac-Citridone A" Org. Lett. 2011, 13, 4592.
10th Most Read Article in Organic Letters: Months September-October
23. T. Cottin, C. Pyrkotis, C. I. Stathakis, I. Mavridis, I. A. Katsoulis, P. Anastasopoulou, G. Kythreoti, A. L. Zografos, V. R. Nahmias, A. Papakyriakou, D. Vourloumis " Designed Spiro-Bicyclic Analogues Targeting the Ribosomal Decoding Center" Chem. Biochem. 2011, 12, 1969.
22. A. L. Zografos "Sommelet-Hauser Rearrangement" Name Reactions in Heterocyclic Chemistry; Chapter 3.11; Editor: J. J. Li; Wiley & Sons 2011.
21. A. L. Zografos "Lehmstedt-Tanasescu Reaction" Name Reactions in Heterocyclic Chemistry; Chapter 7.3; Editor: J. J. Li; Wiley & Sons 2011.
20. I. A. Katsoulis, C. Pyrkotis, A. Papakyriakou, G. Kythreoti, A. L. Zografos, I. Mavridis, V. R. Nahmias, P. Anastasopoulou, Dionisios Vourloumis; "Unnatural Rigid Scaffolds Targeting the Bacterial Ribosome" Chem. Biochem. 2009, 10, 1969.
19. S. A. Snyder, S. P. Breazzano, A. G. Ross, Y. Lin, A. L. Zografos "Synthesis of resveratrol-based natural products" US patent 20100247462, 30 September 2010.
18. S. A. Snyder, S. P. Breazzano, A. G. Ross, Y. Lin, A. L. Zografos; "Achieving synthetic control when Nature abandons selectivity: Total synthesis of all carbogenic complexity within the resveratrol class" J. Am. Chem. Soc. 2009, 131, 1753.
17. S. Snyder, A. L. Zografos, Y. Lin “Total synthesis of resveratrol-based natural products: a chemoselective solution” Angew. Chem. Int. Ed. 2007, 46, 8186.
16. P. Baran, D. O’Malley, A. L. Zografos; “Total Syntheses of pyrole-imidazole alkaloids” J. Am. Chem. Soc. 2007, 129, 4762.
15. A. L. Zografos, D. Georgiadis; “Synthetic strategies towards naturally occurring tetronic acids”, Synthesis 2006, 3157
14. P. Northrop, D. O´Malley, A. Zografos, P. Baran, K. Houk; “The mechanism of vinyl cyclobutane rearrangement of sceptrin to ageliferin and nagelamide E”, Angew. Chem. Int. Ed. 2006, 45, 4126.
13. A. L. Zografos A. Yiotakis, D. Georgiadis; “Rapid access to the tricyclic core of abyssomicins”, Org. Lett., 2005, 7, 4515.
12. L. Zikou, G. Athanasellis, A. Detsi, A. Zografos, C. Mitsos, O. Igglessi-Markopoulou; “A novel short-step synthesis of functionalized 4-hydroxy-2-quinolones using a 1-hydroxybenzotriazole methodology”, Bull. Chem. Soc Jpn. 2004, 77, 1505.
11. P. Baran, D. O’Malley, A. L. Zografos; “Sceptrin as a biosynthetic precursor to complex pyrrole-imidazole alkaloids: The total synthesis of ageliferin” Angew. Chem. Int. Ed. 2004, 43, 2674.
10. P. Baran, A. L. Zografos, D. O’Malley; “Short total synthesis of sceptrin“ J. Am. Chem. Soc. 2004, 126, 3726.
9. C. Mitsos, A. L. Zografos, O. Igglessi-Markopoulou; “An efficient route for the synthesis of 3-aryl quinolin-2-ones with pharmaceutical interest “ J. Org. Chem. 2003, 68, 4567.
8. C. Mitsos, A. L. Zografos, O. Igglessi-Markopoulou; “Synthesis of tetronic acid derivatives from novel active esters of α-hydroxyacids” J. Heterocyclic Chem. 2002, 39, 1201.
7. A. L. Zografos, C. Mitsos, O. Igglessi-Markopoulou; “Chemoselective cyclization of aminonicotinic acid derivatives to 1,8-naphthyridin-2-ones via a potential intramolecular azadiene-ketene electrocyclization reaction” J. Org. Chem. 2001, 66, 4413.
6. A. L. Zografos, PhD Thesis “Study on the synthesis of β-dicarbonyl heterocyclic derivatives” National Technical University of Athens, 2000.
5. C. Mitsos, A. Zografos, O. Igglessi-Markopoulou; “Reactions of N-hydroxysuccinimide esters of anthranilic acids with anions of β-keto esters. A new route to 4-oxo-3-quinolinecarboxylic acid derivatives” Chem. Pharm. Bull. 2000, 48, 211.
4. C. Mitsos, A. L. Zografos, O. Igglessi-Markopoulou; “Regioselective ring opening of malic acid anhydrides by carbon nucleophiles. Application in the synthesis of chiral tetronic acids” J. Org. Chem. 2000, 65, 5852.
3. C. Mitsos, A. L. Zografos, O. Igglessi-Markopoulou; “Synthesis of 3-susbstituted 4-hydroxyquinolin-2-ones via C-acylation reactions of active methylene compounds with functionalized 3,1-benzoxazin-4-ones” Heterocycles 1999, 51, 1543.
2. A. L. Zografos, C. Mitsos, O. Igglessi-Markopoulou; “One-step synthesis for the preparation of quinoline alkaloid analogues” Org. Lett., 1999 1, 1953.
1. A. L. Zografos, C. Mitsos, O. Igglessi-Markopoulou; “A tandem C-acylation-cyclization reaction sequence for the synthesis of new Ν-acyl-3-substituted 1,8-naphthyridine-2,4-diones” Heterocycles 1999, 51, 1609.
Conference Publications
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1. A. Zografos, O. Igglessi-Markopoulou, ‘Synthesis and structural studies of α-substituted 1,8-naphthyridine-2,4-diones with nuclear magnetic resonance spectroscopy’, Book of abstracts “Symposium of Research and Technology” Institute of Physical Chemistry, Athens, Demokritos, 3-5 December 1997, p. 102. 2. A. Zografos, C. Mitsos, O. Igglessi-Markopoulou, Book of abstracts ”1st International Conference of Chemical Societies of Southeastern Countries” Greece Halkidiki June 1998, PO042. 3. C. Mitsos, A. Zografos, O. Igglessi-Markopoulou, Book of abstracts ”1st International Conference of Chemical Societies of Southeastern Countries” Greece Halkidiki June 1998, PO043. 4. C. Mitsos, A. Zografos, O. Igglessi-Markopoulou, ‘C-acylation reaction of β-ketoesters with active esters of anthranicic acid. A new synthetic route of 4-oxo-quinolin-carboxylic acid’, Book of abstracts “Conference on Chemistry Greece-Cyprus Chemistry and Quality Systems in Production and Control” Rodos island, 2-5 September 1999, p. 422. 5. A. Zografos, C. Mitsos, O. Igglessi-Markopoulou, ‘Synthetic studies of 3-alkyl-4-hydroxy- 1,8-naphthyridin-2-ones. A novel method for preparing them.’, Book of abstracts “Conference on Chemistry Greece-Cyprus Chemistry and Quality Systems in Production and Control” Rodos island, 2-5 September 1999, p. 612. 6. A. Zografos, C. Mitsos, O. Igglessi-Markopoulou, ‘One step synthesis for the preparation of quinoline alkaloid analogues’, Book of abstracts ”2nd International Conference of Chemical Societies of Southeastern Countries” Greece Halkidiki 6-9- June 2000, p.152. 7. C. Mitsos, A. Zografos, O. Igglessi-Markopoulou, ‘A new methodology for the synthesis of tetronic acids utilizing novel N-hydroxy-succinimide esters of α-acetoxyacids’, Book of abstracts ” 2nd International Conference of Chemical Societies of Southeastern Countries” Greece Halkidiki 6-9 June 2000, p.158. 8. G. Athanaselis, E. Gavrielatos, A. Zografos, O. Igglessi-Markopoulou, J. Markopoulos, ‘Synthesis, Crystal Structure and Spectral properties of a Copper (II) Complex with N-Acetyl-3-Butanoyl Tetramic Acid‘ Book of abstracts “34th International Conference on Coordination Chemistry” UK, Edinburgh, 9-14 July 2000, PO240. 9. C. Mitsos, A. Zografos, O. Igglessi-Markopoulou, ‘A new simple route to naturally occurring 3-acyl-5-carboxymethyl tetronic acids’ Book of abstracts “7th Sina Conference on Pure and Applied Heterocyclic Chemistry” Egypt, Alexandria, 25-28 March 2000, P-124. 10. A. Zografos, C. Mitsos, O. Igglessi-Markopoulou, ‘One step synthesis for the preparation of quinoline alkaloid analogues’ Book of abstracts “7th Sina Conference on Pure and Applied Heterocyclic Chemistry” Egypt, Alexandria, 25-28 March 2000, P-126. 11. L. Zikou, A. Zografos, ¨Approch to quinoline alkaloid core by the use of silyl ketene acetals¨ “Tetrahedron Symposium” France, Bordeaux, June 2005. 12. A. Zografos, P. Anastasopoulou, A.Yiotakis, D. Georgiadis, ¨Enantioselective synthetic approach to RXPA380¨ “Hellenic Conference” Greece, Ioannina, 20-23 September 2005. 13. A. Zografos, P. Anastasopoulou, A. Yiotakis, D. Georgiadis ¨Stereospecific Synthetic Approach Towards RXPA380, A Potent And Selective Phosphinic Inhibitor Of The C-Domain Of Angiotensin-I Converting Enzyme¨ 5th Hellenic Forum of Bioactive Peptides Greece, Patra 14-16 May 2006. 14. S. Snyder, S. P. Breazzano, A. G. Ross, Y. Lin, A. L. Zografos, ¨Achieving synthetic control when nature abandons selectivity¨ Gordon Research Conference on Natural Products, USA, Tilton, NH, July 2008. 15. A. L. Zografos "Natural Products-Mines of Inspiration" 2nd EUCHEM Conference, Germany, Regensburg, 2010 16. E. E. Anagnostaki, A. L. Zografos Association of Greek Chemists Conference, Greece, Thessaloniki, 2011. 17. A. L. Zografos, STEMCHEM COST-Meeting, 27-28 March 2014, Budapest, Hungary, (Invited presentation) 18. A. L. Zografos, Anatolian Conference of Organic Synthesis, 16-19 March 2015, Antalya, Turkey, (Invited presentation) 19. A. L. Zografos, 12th Greek-Cyprus Conference, 8-10 May 2015, Thessaloniki, Greece (Invited presentation) 20. A. L. Zografos, 9eme Recontres de Chimie Organique de Marseille 9-10 June 2016, Marseille, France (Invited presentation)
21. E. Kontogiannidou, N.
Bouropoulos, D. Andreadis, E. Demiri, A. Zografos, C. Karavasili, D. G.
Fatouros " Permeation enhacement of macromolecules across human skin in
vitro by microneedle device and terpenes" CRS conference
22. A. L.
Zografos, Chemistry at the Interface of Biology and
Medicine, 23-26 September 2016, Heraklion, Crete, Greece (Invited
presentation) 23.
A. L. Zografos,
CHAOS COST-Meeting, 26-29 September 2016, Vienna Austria (Invited
presentation) 24.
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This site was last updated 11-12-2016